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Zaldaride maleate

CAS No.: 109826-27-9

Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity (IC50: 3.3 nM). Zaldaride maleate
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Description Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity (IC50: 3.3 nM). Zaldaride maleate is an effective and selective inhibitor of calmodulin. Zaldaride maleate prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+, and K+ currents in PC12 cells and inhibits nAChR.
Target activity Calmodulin:3.3 nM
Synonyms CGS-9343B, KW 5617
molecular weight 544.6
Molecular formula C30H32N4O6
CAS 109826-27-9
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