Description | Zaldaride maleate inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity (IC50: 3.3 nM). Zaldaride maleate is an effective and selective inhibitor of calmodulin. Zaldaride maleate prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+, and K+ currents in PC12 cells and inhibits nAChR. |
Target activity | Calmodulin:3.3 nM |
Synonyms | CGS-9343B, KW 5617 |
molecular weight | 544.6 |
Molecular formula | C30H32N4O6 |
CAS | 109826-27-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |