| Description | YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki values of 68 pM and 63 nM for CCK-B and CCK-A receptor, respectively. |
| Target activity | CCR2:63 nM （ki）, CCR1:68 pM （ki） |
| molecular weight | 516.59 |
| Molecular formula | C32H28N4O3 |
| CAS | 145084-28-2 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |