| Description | WIN site inhibitor 1 is a WIN site of chromatin-associated WD repeat-containing protein 5 (WDR5) inhibitor (Kd: 0.1 nM), with anti-cancer activity. |
| Target activity | WIN:(kd)0.1 nM |
| Synonyms | WIN site inhibitor 1 |
| molecular weight | 498.38 |
| Molecular formula | C25H22Cl2FN5O |
| CAS | 2407457-36-5 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| References | 1. Aho ER, et al. Displacement of WDR5 from Chromatin by a WIN Site Inhibitor with Picomolar Affinity. Cell Rep. 2019 Mar 12;26(11):2916-2928.e13. |