| Description | VU041 is an inhibitor of Anopheles gambiae and Aedes aegypti inward rectifier potassium 1 channels (IC50: 2.5 μM and 1.7 μM, respectively). VU041 inhibits appreciably is mammalian Kir2.1 (IC50: 12.7 μM) and has less inhibitory effect on mammalian Kir1.1, Kir4.1, Kir6.2/SUR1, and Kir7.1. |
| Target activity | Kir2.1 (mammalian):12.7 μM, Kir1 channel (Anopheles An. gambiae):2.5 μM, Kir1 channel (aedes Ae. aegypti):1.7 μM |
| molecular weight | 363.38 |
| Molecular formula | C19H20F3N3O |
| CAS | 332943-64-3 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |