| Description | Trelagliptin (SYR-472) is a highly specific and long-acting DPP-4 inhibitor. |
| Target activity | DPP4:4 nM (IC50) |
| Synonyms | SYR-472, 曲格列汀 |
| molecular weight | 357.38 |
| Molecular formula | C18H20FN5O2 |
| CAS | 865759-25-7 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility | Ethanol: 3 mg/mL (8.39 mM), Heating is recommended. DMSO: 55 mg/mL (153.9 mM), Sonication is recommended. H2O: < 1 mg/mL (insoluble or slightly soluble) |
| References | 1. Inagaki N, et al. Lancet Diabetes Endocrinol. 2014, 2(2), 125-132. |