| Description | TCS PIM-1 1 (SC 204330)(sc-204330) is a effective and specific ATP-competitive Pim-1 kianse inhibitor (IC50: 50 nM) , exhibits good specific over MEK1/MEK2 and Pim-2(IC50s >20, 000 nM). |
| Target activity | Pim1:50 nM |
| Synonyms | 3-氰基-4-苯基-6-(3-溴-6-羟基苯基)-2(1H)-吡啶酮, SC 204330 |
| molecular weight | 367.2 |
| Molecular formula | C18H11BrN2O2 |
| CAS | 491871-58-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| Solubility | DMSO: 16.67 mg/mL (45.39 mM), Sonication is recommended. |
| References | 1. Cheney IW, et al. Bioorg Med Chem Lett. 2007 Mar 15;17(6):1679-83. |