| Description | TAP311 is an inhibitor of cholesteryl ester transfer protein (CETP)(IC50 of 62 nM). |
| Target activity | CETP:62 nM |
| molecular weight | 710.71 |
| Molecular formula | C34H40F6N6O4 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| References | 1. Yamada K, et al. Discovery of a Novel Piperidine-Based Inhibitor of Cholesteryl Ester Transfer Protein (CETP) That Retains Activity in Hypertriglyceridemic Plasma. J Med Chem. 2017 Oct 26;60(20):8466-8481. |