| Description | PF-4136309 (INCB8761, PF-04136309) is a highly effective and selective oral CCR2 antagonist with good bioavailability, with an IC50 value of 5.2 nM for human CCR2. |
| Target activity | CCR2:5.2 nM |
| Synonyms | PF-04136309, INCB8761 |
| molecular weight | 568.59 |
| Molecular formula | C29H31F3N6O3 |
| CAS | 857679-55-1 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| References | 1. Xianming Deng, et, al. Eur J Med Chem. 2013;70:758-67. 2. Xue CB, et al. ACS Med Chem Lett. 2011 Oct 5;2(12):913-8. |
(Rac)-PF-4136309（1341224-83-6 Free base)
CAS No.: 857679-55-1
PF-4136309 (INCB8761, PF-04136309) is a highly effective and selective oral CCR2 antagonist with good bioavailability, w
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