| Description | PI3Kdelta inhibitor 1 is a potent, selective and orally available inhibitor of PI3Kδ with an IC50 of 1.3 nM. |
| Target activity | PI3Kδ:1.3 nM |
| molecular weight | 558.69 |
| Molecular formula | C27H38N6O5S |
| CAS | 2242109-74-4 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| References | 1. Hamajima T, et al. Optimization and in vivo evaluation of pyrazolopyridines as a potent and selective PI3Kδ inhibitor. Bioorg Med Chem. 2018 Aug 7;26(14):3917-3924. |