| Description | PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist. |
| Target activity | OTR:9.5 nM |
| Synonyms | PF 3274167, Cligosiban, PF-3274167 |
| molecular weight | 419.84 |
| Molecular formula | C19H19ClFN5O3 |
| CAS | 900510-03-4 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| Solubility | DMSO: 55 mg/mL (131 mM), Sonication is recommended. |
| References | 1. Karpenko IA, et al. J Med Chem. 2015 Mar 12;58(5):2547-52. 2. Brown A, et al. Bioorg Med Chem Lett. 2010 Jan 15;20(2):516-20. |