| Description | Molibresib besylate is an inhibitor of BET bromodomain (IC50: 32.5-42.5 nM). |
| Target activity | BET:32.5-42.5 nM |
| Synonyms | I-BET 762 besylate, GSK 525762C |
| molecular weight | 582.07 |
| Molecular formula | C28H28ClN5O5S |
| CAS | 1895049-20-3 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| Solubility | DMSO: 25 mg/mL (42.95 mM), Sonication is recommended. |
| References | 1. Nicodeme E, et al. Suppression of inflammation by a synthetic histone mimic. Nature. 2010 Dec 23;468(7327):1119-23. |