| Description | ML230 is a selective ATP-binding cassette (ABC) transporter ABCG2 inhibitor. It 36-fold selective for ABCG2 over ABCB1 (EC50s: 0.13 μM and 4.65 μM, respectively). |
| Target activity | ABCG2:0.13 μM(EC50) |
| Synonyms | CID44640177, SID 88095709 |
| molecular weight | 439.47 |
| Molecular formula | C25H21N5O3 |
| CAS | 1776055-05-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| References | 1. Strouse JJ, et al. Selective Efflux Inhibition of ATP-binding Cassette Sub-family G Member 2. Probe Reports from the NIH Molecular Libraries Program. November 30, 2010. |