| Description | Lomitapide Mesylate (BMS-201038 mesylate) is a methanesulfonic acid form of lomitapide, a small molecule inhibitor of microsomal triglyceride transfer protein. |
| Target activity | MTP:8 nM |
| Synonyms | 甲磺酸洛美他派, BMS-201038 mesylate, AEGR-733 mesylate |
| molecular weight | 789.83 |
| Molecular formula | C40H41F6N3O5S |
| CAS | 202914-84-9 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| Solubility | H2O: < 1 mg/mL (insoluble or slightly soluble) Ethanol: 93 mg/mL (117.7 mM) DMSO: 93 mg/mL (117.7 mM) |
| References | 1. Davis KA, Miyares MA. Am J Health Syst Pharm. 2014 Jun 15;71(12):1001-8. |