| Description | KS176 is a potent and selective inhibitor of the breast cancer resistance protein (BCRP) multidrug transporter, showing no inhibitory activity against P-gp or MRP1. |
| Target activity | BCRP(Pheo A):0.59 μM |
| molecular weight | 405.4 |
| Molecular formula | C22H19N3O5 |
| CAS | 1253452-78-6 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| Solubility | DMSO: 55 mg/mL (135.67 mM) |
| References | 1. Pick A, et al. Specific inhibitors of the breast cancer resistance protein (BCRP). ChemMedChem. 2010 Sep 3;5(9):1498-505. |