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JTZ-951 HCl

CAS No.: 1262131-60-1

JTZ-951 is a potent and orally active inhibitor of hypoxia inducible factor prolyl hydroxylase (PHD).
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Description JTZ-951 is a potent and orally active inhibitor of hypoxia inducible factor prolyl hydroxylase (PHD).
Synonyms JTZ-951, JTZ 951 hydrochloride, JTZ951 HCl, JTZ 951
molecular weight 376.79
Molecular formula C17H17ClN4O4
CAS 1262131-60-1
Storage Powder: -20°C for 3 years | In solvent: -80°C for 1 year
References 1. Discovery of JTZ-951: A HIF Prolyl Hydroxylase Inhibitor for the Treatment of Renal Anemia Yosuke Ogoshi, Takuya Matsui, Ikuo Mitani, Masahiro Yokota, Masakazu Terashita, Dai Motoda, Kazuhito Ueyama, Takahiro Hotta, Takashi Ito, Yasunori Hase, Kenji Fukui, Katsuya Deai, Hiromi Yoshiuchi, Soichiro Ito, and Hiroyuki Abe Publication Date (Web): November 20, 2017 (Letter) doi: 10.1021/acsmedchemlett.7b00404