Description | EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5). |
Target activity | EP1:7.54(pKi), EP1:8.5(pIC50) |
Synonyms | EP1-antanoist-1, EP1 antagonist 1 |
molecular weight | 470.14 |
Molecular formula | C19H15BrCl2N2O3 |
CAS | 851204-35-8 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
Solubility | DMSO: 55 mg/mL (116.99 mM) |
References | 1. eown SC, et al. Identification of novel pyrazole acid antagonists for the EP1 receptor. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4767-7Epub 2006 Jul 14. |