| Description | Enpp-1-IN-17 (example 274) is a potent inhibitor of ENPP1, exhibiting inhibition constants (Ki values) of 100 nM-1 μM for cGAMP hydrolysis and >1 μM for ATP hydrolysis, respectively, with a selectivity ratio of >6.4 favoring cGAMP hydrolysis inhibition [1]. |
| molecular weight | 328.41 |
| Molecular formula | C18H24N4O2 |
| CAS | 2289736-54-3 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |