| Description | DDPM-2571 is a highly potent and in vivo active inhibitor of GABA transporter subtype 1 with anticonvulsant, anxiolytic, antidepressant and antinociceptive properties. DDPM-2571 was quickly distributed into the brain and was highly effective in the prevention of chemically-induced seizures (pentylenetetrazole and pilocarpine models) and 6-Hz convulsions. It demonstrated significant anxiolytic-like and antidepressant-like properties. DDPM-2571 had antinociceptive properties, both in the hot plate test and in the second phase of the formalin test. |
| molecular weight | 455.76 |
| Molecular formula | C21H21Cl3N2O3 |
| CAS | 1672672-26-2 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |