| Description | CPI-169 (R) is a novel and potent inhibitor of EZH2. |
| Target activity | EZH2 (Y641N):0.51 nM (IC50), EZH2 (WT):0.24 nM (IC50), EZH1:6.1 nM (IC50) |
| Synonyms | CPI 169 (R), CPI-169 (R) |
| molecular weight | 528.66 |
| Molecular formula | C27H36N4O5S |
| CAS | 1802175-07-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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