PeptideDB

CGP 64213

CAS No.: 200402-50-2

CGP 64213 is a GABAb receptor agonist.
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Description CGP 64213 is a GABAb receptor agonist.
Synonyms CGP-64213, CGP64213
molecular weight 646.45
Molecular formula C26H36IN2O7P
CAS 200402-50-2
Storage Powder: -20°C for 3 years | In solvent: -80°C for 1 year
References 1. Duthey B, Caudron S, Perroy J, Bettler B, Fagni L, Pin JP, Prézeau L. A single subunit (GB2) is required for G-protein activation by the heterodimeric GABA(B) receptor. J Biol Chem. 2002 Feb 1;277(5):3236-41. PubMed PMID: 11711539; PubMed Central PMCID: PMC2566549. 2. Calon F, Lavertu N, Lemieux AM, Morissette M, Goulet M, Grondin R, Blanchet PJ, Bédard PJ, Di Paolo T. Effect of MPTP-induced denervation on basal ganglia GABA(B) receptors: correlation with dopamine concentrations and dopamine transporter. Synapse. 2001 Jun 1;40(3):225-34. PubMed PMID: 11304760. 3. Calon F, Morissette M, Goulet M, Grondin R, Blanchet PJ, Bédard PJ, Di Paolo T. 125I-CGP 64213 binding to GABA(B) receptors in the brain of monkeys: effect of MPTP and dopaminomimetic treatments. Exp Neurol. 2000 May;163(1):191-9. PubMed PMID: 10785458. 4. Froestl W, Bettler B, Bittiger H, Heid J, Kaupmann K, Mickel SJ, Strub D. Ligands for the isolation of GABA(B) receptors [corrected] . Neuropharmacology. 1999 Nov;38(11):1641-6. Review. Erratum in: Neuropharmacology 1999 Dec;38(12):1921. PubMed PMID: 10587079.