| Description | CB1/2 agonist 1 is a potent CB1/2 agonist that crosses the blood-brain barrier, acting on CB1R (EC50: 56.15 nM) and CB2R (EC50: 11.63 nM). CB1/2 agonist 1 reduces glutamate release and LPS-induced microglia activation, and has anti-inflammatory and analgesic activities. CB1/2 agonist 1 has potential for multiple sclerosis studies. |
| molecular weight | 435.33 |
| Molecular formula | C21H24BrFN2O2 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |