PeptideDB

BM213

CAS No.: 2891606-02-1

BM213是一种选择性的C5aR1激动剂,EC50为59 nM,可诱导C5aR1介导的钙动员和pERK1/2信号通路,但不能诱导β-抑制素的募集。BM213
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Description BM213是一种选择性的C5aR1激动剂,EC50为59 nM,可诱导C5aR1介导的钙动员和pERK1/2信号通路,但不能诱导β-抑制素的募集。BM213更为稳定,对SHSY-5Y 细胞无细胞毒性。
Synonyms BM213
molecular weight 915.09
Molecular formula C43H70N12O10
CAS 2891606-02-1
Storage keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year
References 1. Gorman DM, et al. J Med Chem. 2021 Nov 25;64(22):16598-16608.