| Description | Bisubstrate Inhibitor 78 HCl is an NNMT inhibitor (IC50 = 1.41 μM) with potential anticancer activity, inhibiting the proliferation of HSC-2 oral cancer cells at 100 μM. |
| Synonyms | Bisubstrate Inhibitor 78 HCl(2368247-39-4 Free base) |
| molecular weight | 544 |
| Molecular formula | C25H30ClN7O5 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| References | 1. Gao Y,et al. Bisubstrate Inhibitors of Nicotinamide N-Methyltransferase (NNMT) with Enhanced Activity. J Med Chem. 2019 Jul 25;62(14):6597-6614. |