Description | ARDP0006 is an inhibitor of NS2B-NS3 protease. |
Synonyms | 1,8-二羟基-4,5-二硝基蒽醌 |
molecular weight | 330.21 |
Molecular formula | C14H6N2O8 |
CAS | 81-55-0 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Solubility | DMSO: Slightly soluble |
References | 1. Justin Jang Hann Chu, Regina Ching Hua Lee, Melgious Jin Yan Ang,et al.Antiviral activities of 15 dengue NS2B-NS3 protease inhibitors using a human cell-based viral quantification assay.Antiviral Res. 2015 Jun;118:68-74. doi: 10.1016/j.antiviral.2015.03.010. Epub 2015 Mar 27. 2. Constant D A , Mateo R , Nagamine C M , et al. Targeting intramolecular proteinase NS2B/3 cleavages for trans -dominant inhibition of dengue virus[J]. Proceedings of the National Academy of Sciences, 2018, 115(40):201805195. |