| Description | Acetyl-Calpastatin (184-210)(human) acetate is a potent, selective and reversible calpain inhibitor with Ki values of 0.2 nM and 6 μM for µ-calpain and cathepsin L, respectively. |
| In vitro | Acetyl-Calpastatin (184-210)(human) acetate (peptide 1; 12.5-100 μM) 在 LCLC 103H 细胞中抑制 calpains，其 IC50 为 27 μM[1]。 |
| Synonyms | Acetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base ) |
| molecular weight | 3237.68 |
| Molecular formula | C144H234N36O46S |
| Storage | store at low temperature,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| References | 1. Ferdinando Fiorino, et al. A new cell-permeable calpain inhibitor. J Pept Sci. 2007 Jan;13(1):70-3. 2. Benjamin P Davis, et al. Eosinophilic esophagitis-linked calpain 14 is an IL-13-induced protease that mediates esophageal epithelial barrier impairment. JCI Insight. 2016 Apr;1(4):e86355. |
Acetyl-Calpastatin (184-210)(human) acetate
CAS No.:
Acetyl-Calpastatin (184-210)(human) acetate is a potent, selective and reversible calpain inhibitor with Ki values of 0.
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