Description | Guvacine can enhance the inhibition of spinal neurones by GABA. |
Target activity | GAT-1 (rat):39 μM (IC50), GAT-2 (rat):58 μM (IC50), GAT-1 (human):14 μM (IC50), GAT-3 (human):119 μM (IC50), BGT3 (human):1870 μM (IC50), GAT-3 (rat):378 μM (IC50) |
molecular weight | 127.14 |
Molecular formula | C6H9NO2 |
CAS | 498-96-4 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |