Bioactivity | Parapenzolate bromide, an antispasmodic, is an orally active mAChR antagonist. Parapenzolate bromide is an anticholinergic agent[1][2]. |
In Vivo | Parapenzolate bromide (10 mg/kg, p.o. or i.v.) shows a significant analgesic effect in mice[1].Parapenzolate bromide (0.5 mg/kg, i.v.) exhibits a spasmolytic activity in isolated gall bladder from guinea pigs[2]. Animal Model: |
Name | Parapenzolate bromide |
CAS | 5634-41-3 |
Formula | C21H26BrNO3 |
Molar Mass | 420.34 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Paris, J., et al. Effect of parapenzolate bromide on the contractility of the gall bladder and sphincter of Oddi. Therapie (1968), 23(3), 609-18. [2]. Ishimura Yasuko, et al. Pharmacological studies on parapenzolate bromide. 1. Pharmacological studies. Shikoku Igaku Zasshi (1970), 26(1), 43-51. |