| Bioactivity | GPR109 receptor agonist-1 (Compound 3a) is a highly selective agonist of the human orphan G-protein-coupled receptor GPR109b, with the pEC50 of 6.4. GPR109 receptor agonist-1 can be used for the research of cardio-metabolic diseases[1]. | ||||||||||||
| Target | pEC50: 6.40 ± 0.36 (GPR109b) | ||||||||||||
| Name | GPR109 receptor agonist-1 | ||||||||||||
| CAS | 306935-41-1 | ||||||||||||
| Formula | C10H11N3O2 | ||||||||||||
| Molar Mass | 205.21 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
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| Reference | [1]. Graeme Semple, et al. 1-Alkyl-benzotriazole-5-carboxylic acids are highly selective agonists of the human orphan G-protein-coupled receptor GPR109b. J Med Chem. 2006 Feb 23;49(4):1227-30. |
GPR109 receptor agonist-1
CAS: 306935-41-1 F: C10H11N3O2 W: 205.21
GPR109 receptor agonist-1 (Compound 3a) is a highly selective agonist of the human orphan G-protein-coupled receptor GPR
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