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Bioactivity FGH31 (Compound 24) is a potent, selective, GRK2 dependency dopamine D4 agonist, with the Ki of 1.6 nM. FGH31 partial activates β- arrestin[1].
Invitro FGH31 (Compound 24) (50 μM) 在大鼠肝微粒体中的下降速率与 Imipramine (HY-B1490A) 相似[1]。FGH31 (50 μM, 4 h) 在 Caco-2 细胞中未发生 p -糖蛋白 (P-gp) 介导的转运[1]。 0 --> FGH31 相关抗体:
Name FGH31
Formula C33H36N4O2
Molar Mass 520.66
Transport Room temperature in continental US; may vary elsewhere.

Please store the product under the recommended conditions in the Certificate of Analysis.

Reference [1]. Graßl F, et al. Exploring Structural Determinants of Bias among D4 Subtype-Selective Dopamine Receptor Agonists. J Med Chem. 2023;66(14):9710-9730. doi:10.1021/acs.jmedchem.3c00537

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